Aspirin UPSA: malangizo ogwiritsira ntchito

Kutulutsa Fomu

Mphamvu za miyala yozungulira yozungulira, yoyera. Akasungunuka m'madzi, amadzimadzi a gasi amamasulidwa.

Zogwira pophika: acetylsalicylic acid (500 mg), zotulutsa: sodium carbonate anhydrous, citric acid anhydrous, sodium citrate anhydrous, sodium bicarbonate, crospovidone, aspartame, kuwala kwachilengedwe kwa lalanje, povidone.

Vitamini C: acetylsalicylic acid (330 mg), ascorbic acid (200 mg). Omwe amathandizira: glycine, sodium benzoate, anhydrous citric acid, monosodium carbonate, polyvinylpyrrolidone.

4 mapiritsi amagetsi mu mzere wa zotayidwa zojambulazo zokutira mkati ndi polyethylene. Mzere 4 kapena 25 pamodzi ndi malangizo ogwiritsira ntchito paketi yamakhadi.

Vitamini C: Mapiritsi 10 pa chubu limodzi. Mmodzi kapena awiri machubu okhala mu katoni

Zotsatira za pharmacological

Ili ndi anti-yotupa, analgesic komanso antipyretic zotsatira zoyenderana ndi kuponderezana kwa cycloo oxygenase 1 ndi 2, kuyang'anira kapangidwe ka prostaglandins. Amachepetsa kusakanikirana, kuphatikizika kwa mapulateleti ndi thrombosis mwa kupondereza kaphatikizidwe ka thromboxane A2 m'maselo, pomwe mphamvu ya antiplatelet imapitilira sabata pambuyo pa limodzi.

Ubwino wa mtundu wosungunuka wa mankhwala poyerekeza ndi miyambo ya acetylsalicylic acid m'mapiritsi ndi njira yomaliziratu komanso yogwira ntchito mwachangu.

Pharmacokinetics

UPSA aspirin imamwidwa mwachangu kuposa aspirin wokhazikika. Kuchuluka kwa acetylsalicylic acid kumafikira mphindi 20. The plasma theka moyo ndi kuyambira 15 mpaka 30 mphindi. Acetylsalicylic acid imadutsa hydrolysis mu plasma ndi mapangidwe a salicylic acid. Salicylate imagwirizanitsidwa kwambiri ndi mapuloteni a plasma. Kuchiritsa kwa urin kumatuluka ndi mkodzo pH. Hafu ya moyo wa salicylic acid imayambira maola atatu mpaka 9 ndikuwonjezeka ndi kumwa.

  • Kupweteka kwapang'onopang'ono kapena kofatsa mwa achikulire osiyanasiyana komwe kumachokera: mutu wambiri (kuphatikizapo omwe amaphatikizidwa ndi vuto lodziletsa zakumwa zoledzeretsa), mano, migraine, neuralgia, radicular radicular syndrome, kupweteka kwa minofu ndi kuphatikizana, kupweteka pakapita msambo.
  • Kuchuluka kwa kutentha kwa thupi kuzizira ndi matenda ena opatsirana komanso otupa (mwa akulu ndi ana opitilira zaka 15).

Contraindication

  • Zilonda zam'mimba komanso zam'minyewa zam'mimba.
  • Matenda oopsa a portal,
  • "Aspirin" mphumu,
  • Exortating Aortic Aneurysm,
  • Phenylketonuria,
  • Hemorrhagic diathesis, kuphatikizapo hemophilia, telangiectasia, matenda a Willebrand, thrombocytopenia, hypoprothrombinemia, thrombocytopenic purpura,
  • Glucose-6-phosphate dehydrogenase akusowa,
  • Hypersensitivity pamagawo a Aspirin UPSA kapena mankhwala ena osapweteka a antiidal
  • Kuopsa kwa chiwindi ndi impso.
  • Kuperewera kwa Vitamini K

Mankhwalawa amaloledwa kumwa kokha mwa II trimester ya kutenga pakati, pamene amwedwa panthawi ya mkaka wa m'mawere, kuyamwitsa kumalimbikitsidwa. Aspirin UPSA sagwiritsidwa ntchito mwa ana ochepera zaka 15 chifukwa cha vuto la Reye syndrome.

Aspirin ayenera kumwedwa. ndi chisamaliro ndi urate nephrolithiasis, hyperuricemia, mtima kuwonda ndi zilonda zam'mimba ndi duodenum mu anamnesis. Mukamagwiritsa ntchito aspirin, ziyenera kukumbukiridwa kuti zingayambitse kugunda kwamatenda kwa gout ndi vuto lomwe lidalipo kale.

Mlingo ndi makonzedwe

Mlingo ndi ndandanda ya kuvomerezedwa imatsimikiziridwa ndi adotolo, chifukwa pano zonse zimatengera zaka komanso momwe wodwalayo alili.

Mapiritsi a mphamvu a ngokuyambirira ayenera kusungunuka mu 100-200 mg ya madzi owiritsa firiji. Mankhwala ayenera kumwedwa mutatha kudya.

Ndi ululu waukulu, mutha kutenga 400-800 mg ya acetylsalicylic acid katatu patsiku (koma osapitirira 6 g patsiku). Monga othandizira antiplatelet, milingo yaying'ono imagwiritsidwa ntchito - 50, 75, 100, 300 kapena 325 mg pazinthu zomwe zikugwira ntchito. Pa malungo, tikulimbikitsidwa kuti muthe kutenga 0,5-1 g wa acetylsalicylic acid patsiku (ngati kuli kotheka, mlingowo utha kuwonjezeka mpaka 3 g).

Kutalika kwa chithandizo sikuyenera kupitilira masiku 14.

Zotsatira zoyipa

Mlingo wovomerezeka, Aspirin UPSA nthawi zambiri imalekeredwa. Nthawi zambiri, mukamwa mankhwalawa, mavuto otsatirawa akhoza kukhala:

  • Khungu, "pririn triad", bronchospasm ndi edincke's,
  • Matenda a impso,
  • Epistaxis, nthawi yochulukitsa, zotulutsa magazi,
  • Kuchepetsa mseru, kuchepa kwa chilala, kusanza, kutaya m'mimba, kupweteka kwam'mimba, kutsekula m'mimba,
  • Supombocytopenia, leukopenia, kuchepa magazi, hyperbilirubinemia.

Zotsatira zosafunikira zikachitika, makonzedwe a Aspirin UPSA ayenera kusiyidwa.

Bongo

Muyenera kusamala ndi kuledzera kwa okalamba makamaka ana aang'ono (mankhwala osokoneza bongo kapena kuledzera mwangozi, omwe amapezeka nthawi zambiri mwa ana aang'ono kwambiri), omwe angayambitse imfa.

Zizindikiro zamankhwala - ndi kuledzera koyenera, tinnitus ndiyotheka, kusamva kwa mutu, kupweteka mutu, chizungulire, nseru ndi chizindikiro cha bongo. Izi zimachotsedwa pochepetsa mlingo. Kuledzera kwambiri - hyperventilation, ketosis, kupumula kwa alkalosis, metabolic acidosis, chikomokere, kugwa kwa mtima, kulephera kupuma, kuchepa kwapafupipafupi.

Chithandizo - Kuchotsa mwachangu mankhwalawa posambitsa m'mimba. Kugonekedwa kuchipatala kwapadera. Acid-base balance control. Kukakamizidwa zamchere diuresis, hemodialysis, kapena peritoneal dialysis ngati pakufunika.

Kuyanjana kwa mankhwala osokoneza bongo

Kuphatikiza kwa methotrexate kumatsutsana, makamaka pamtunda waukulu (izi zimawonjezera kawopsedwe), ndikamayamwa anticoagulants pamtunda waukulu, chiopsezo cha magazi chikuwonjezeka.

Kuphatikiza kosafunikira - ndi ma anticoagulants am'mlomo (pamiyeso yotsika, chiopsezo chotulutsa magazi), ndi ticlopidine (kumawonjezera chiopsezo cha magazi), ndi ma uricosuric othandizira (kuchepa kwa mphamvu ya uricosuric ndikotheka), ndi mankhwala ena odana ndi kutupa.

Kuphatikiza komwe kumafunikira kusamala: ndi antidiabetesic othandizira (makamaka, kuchepetsa sulfamides) - kuchuluka kwa hypoglycemic kumakulirakulira, ma antacid - nthawi zopitilira pakati pa ma antacid ndi mankhwala a salicylic uyenera kuchitika (maola 2), ndi okodzetsa - okhala ndi mankhwala okwanira Madzi, yang'anirani ntchito ya impso kumayambiriro kwa chithandizo chifukwa chotheka kupweteka kwaimpso kwa wodwala wopanda madzi, wokhala ndi corticoids (glucocorticoids) ) - mwina ndichepe salitsilemii pa mankhwala ndi corticoids ndipo pali chiopsezo kuti ambiri osokoneza wa salicylate pambuyo kuchotsa ake.

Mimba komanso kuyamwa

Mankhwala ndi contraindicated pa mimba mu I ndi III trimester. Munthawi yachiwiri yomwe mayi ali ndi pakati, kumwa limodzi mwa mankhwalawa komwe kungatheke. Ngati kuli kofunikira kugwiritsa ntchito mankhwalawa panthawi yoyamwitsa, kuyamwa kuyenera kuyimitsidwa.

Malangizo apadera

Mankhwalawa amatha kuthandizira kutaya magazi, komanso kuonjezera nthawi ya msambo. Aspirin imakulitsa chiopsezo chotaya magazi ngati angachitidwe opareshoni.

Mu ana, popanga mankhwala, muyenera kuganizira zaka ndi kulemera kwa thupi.

Ndi zakudya zopanda mchere, popanga zakudya za tsiku ndi tsiku, ziyenera kukumbukiridwa kuti piritsi lililonse la UPSA aspirin wokhala ndi vitamini C lili ndi 485 mg wa sodium.

Mu nyama, teratogenic mphamvu ya mankhwala imadziwika.

Zizindikiro zogwiritsidwa ntchito

Malinga ndi malangizo, Aspirin Oops akuwonetsedwa:

  • Matenda ozizira, opatsirana komanso otupa mwa ana opitilira zaka 15 ndi akulu, omwe amatsagana ndi malungo.
  • Kupweteka kwapang'onopang'ono kapena kwapakati kwa odwala akuluakulu omwe ali ndi magawo osiyanasiyana: kupweteka mutu, kuledzera, migraine, mano, chifuwa cha radicular syndrome, neuralgia, algomenorrhea, kupweteka kwa minofu ndi minyewa.

Mlingo ndi makonzedwe

Mapiritsi Aspirin Oops musanagwiritse ntchito ayenera kusungunuka mu theka kapu ya madzi kapena madzi.

Ana opitirira zaka 15 ndi odwala achikulire amapatsidwa piritsi limodzi mpaka 6 pa tsiku. Ndi kupweteka kwambiri, kutentha kwambiri, kukhazikika kwa Aspirin Ups amaloledwa mu mapiritsi awiri. Mulingo wambiri watsiku ndi tsiku sayenera kupitilira mapiritsi 6 (3 g).

Okalamba odwala Aspirin Ups ndi mankhwala piritsi limodzi mpaka 4 pa tsiku. Kuwona pafupipafupi njira ya kagwiritsidwe ntchito ka Aspirin Oops kumakupatsani mwayi wochepetsera kupweteka kwa ululu komanso kupewa kuwonjezeka kwa kutentha kwa thupi.

Kutalika kwa mankhwalawa sikuyenera kupitirira masiku 5 mutagwiritsidwa ntchito ngati mankhwala oletsa kupweteka komanso masiku atatu ngati antipyretic.

Kugwiritsa ntchito mankhwalawa muyezo waukulu kwa nthawi yayitali kungayambitse zizindikiro zotsatirazi:

  • Mutu wowawa
  • Chizungulire
  • Kumva kutayika,
  • Kupititsa patsogolo
  • Kusanza, kusanza,
  • Zowonongeka
  • Kuponderezedwa kwa chikumbumtima
  • Kuphwanya mphamvu zamagetsi zamagetsi,
  • Kulephera kopindulitsa.

Ngati mankhwala osokoneza bongo amachitika, wodwalayo ayenera kusanza kapena kutsuka m'mimba, kumwa adsorbents ndi mankhwala ofewetsa tuvi tolimba. Ndikulimbikitsidwa kupita kuchipatala.

Zotsatira zoyipa

Kugwiritsa ntchito kwa Aspirin Oops kungayambitse zotsatirazi:

  • Allergies: zotupa pakhungu, bronchospasm, edi ya Quincke, "aspirin" triad (mphumu ya bronchial, polyposis ya mphuno ndi mafinya amkati, tsankho la acetylsalicylic acid,
  • Mitsempha yamadzimadzi: kuwonongeka kwa impso,
  • Matumbo a pakhungu: nseru, kusanza, kutsegula m'mimba, kupweteka kwa m'mimba, magazi am'mimba, kuchuluka kwa michere ya chiwindi, kuchepa kwa chilimbikitso,
  • Hematopoietic dongosolo: kuchepa magazi, thrombocytopenia, hyperbilirubinemia, leukopenia,
  • Momwe magazi amapangidwira: hemorrhagic syndrome (kutulutsa magazi m'magazi, mphuno), nthawi yowonjezera magazi.

Pakukula kwa mavuto, wodwalayo ayenera kusiya kutenga Aspirin Ups.

Aspirin UPSA

Malangizo ogwiritsira ntchito:

Aspirin UPSA ndi mankhwala osagwiritsa ntchito mankhwala osokoneza bongo omwe amagwiritsidwa ntchito pothandiza kuchepetsa ululu komanso kuchepetsa kutentha kwa thupi mu matenda otupa kapena opatsirana.

Migwirizano ndi magwiritsidwe akusungidwa

UPSA aspirin, malinga ndi malangizo, iyenera kusungidwa mu mpweya wokwanira, kunja kwa ana ndikutetezedwa ku kuwala, malo owuma, kutentha osapitirira 30 ° C.

Mankhwalawa amawachotsa ku pharmacies popanda mankhwala, moyo wake wa alumali, malinga ndi malingaliro omwe wopanga ali ndi zaka zitatu. Tsiku lotha litatha, malonda ake ayenera kutayidwa.

Kodi mwapeza cholakwika m'mawuwo? Sankhani ndikusindikiza Ctrl + Lowani.

The zikuchokera mankhwala

Zomwe zimagwira zomwe zimatsimikizira kuti mankhwalawa ndi acetylsalicylic acid, zili 500 mg.

Zosakaniza zothandiza zomwe zimapangitsa kapangidwe ka zinthu zomwe zimagwiritsidwa ntchito pochiritsa ndi citric acid, mankhwala ena a sodium (carbonate ndi citrate), kununkhira ndi kununkhira kwa lalanje, aspartame, croslovidone, ndi zina.

Kuchiritsa katundu

Aspirin mu mapiritsi am'madzi amamwa mwachangu kuposa mankhwala omwewo, koma mwanjira yake. Yoyeserera kwambiri m'magazi imapangidwa mphindi 10 mpaka 40 pambuyo pa kuperekedwa. Chomwe chimagwira ndi hydrolyzed kuti chipange salicylic acid, yemwenso imathandizira. Zinthu zonsezi zimafalikira thupi lonse, kuthana ndi zotchinga, zotulutsidwa mkaka.

Acetylsalicylic acid amasandulika m'chiwindi, metabolites ake amuchotsa mkodzo.

Kutulutsa Mafomu

Mtengo wapakati ndi ma ruble 187.

Aspirin amapangidwa mwa mawonekedwe a mapiritsi a effeedcent. Mapiritsi ndi lathyathyathya-cylindrical, ali ndi chamfer komanso chiopsezo chogawana. Mapiritsi atasungunuka, zimachitika ndi kutulutsa kaboni dayokisaidi.

Chogulikacho chimadzaza matuza 4 mapiritsi, pamakatoni 4 - mizere 4, motsatana.

M'mimba komanso HB

Kukonzekera ndi acetylsalicylic acid sikungagwiritsidwe ntchito nthawi imeneyi, makamaka kwa azimayi omwe ali mu 1st kapena 2 thimester, chifukwa choopsa chachikulu cha fetal pathologies (cleft palate, kukhumudwa kwa mapangidwe a mtima). Ngati pakufunika thandizo mwachangu, Mlingo wake uyenera kukhala wocheperako, ndipo phwando liyenera kukhala lalifupi, loyenera kuyang'aniridwa ndi udokotala.

Mu 3 trimester, asidi amatsutsana mwapadera, chifukwa zimatha kuyambitsa kuchuluka kwa fetal, kusagwira ntchito bwino, ntchito yaimpso mwa mwana, mpaka kukulira kulephera.

Kuphatikiza apo, asidi amatha kupangitsa kuti mayi atulutsidwe magazi ndikutalika kwa mayi kapena mwana wosabadwa. Komanso, Mlingo wocheperako wa aspirin nawonso umayambitsa. Mlingo waukulu wa asidi womwe umagwiritsidwa ntchito kumapeto kwa pakati kumayambitsa kukhazikika kwa magazi. Makanda obadwa asanakwane amakonda kwambiri izi.

Amayi okhala ndi mkaka amayeneranso kusiya Aspirin Oops, popeza acetylsalicylic acid imatha kulowa mkaka.

Njira zopewera kupewa ngozi

Ndi njira yayitali ya Aspirin Oops, pamafunika kuchita magazi mwatsatanetsatane ndi magazi, kuwona momwe chiwindi chilili.

  • Odwala omwe ali ndi gout, mankhwalawa amatha kuyambitsa, chifukwa cha kuthekera kwa acetylsalicylic acid poletsa kwamkodzo potulutsa.
  • Odwala omwe akuchitidwa opaleshoni amasiya kuti achepetse magazi nthawi yayitali komanso atatha kulowererapo.
  • Anthu omwe amawongolera kudya kwamchere ayenera kukumbukira kuti ilipo pakupanga kwa Aspirin Oops.

Kuchita mankhwala osokoneza bongo

Ngati pakufunika mankhwala ena, njira ya Aspirin Ups iyenera kuchitika mosamala, popeza acetylsalicylic acid imakumana ndi zigawo zake, zosokoneza malowa. Chifukwa chake, ndikofunikira kudziwitsa dokotala za ndalama zomwe zatengedwa.

  • Aspirin imakulitsa mphamvu za antidiabetesic ndi anticonvulsants, okodzetsa.
  • Mukaphatikizidwa ndi mankhwala omwe ali ndi mowa kapena mowa, kuwonongeka kwa mucous m'mimba, kumatulutsa mphamvu komanso kutalika kwa magazi mkati.
  • Aspirin sangathe kugwiritsidwa ntchito ndi anticoagulants pamlomo, chifukwa cha kufooka kwa mphamvu yotsirizira komanso chiwopsezo chotaya magazi. Ngati ndi kotheka, muyenera kuwunika nthawi zonse kuchuluka kwa magazi.
  • Kukonzekera komwe kumakhala ndi mankhwala a magnesium, aluminium, mchere wa calcium, imathandizira kuchoka kwa salicylates.

Zotsatira zoyipa

Kutengera Mlingo woyendetsedwa ndi opanga kapena madokotala, zotsatira zoyipa sizimakhalapo, koma sizimaphatikizidwa:

  • Mawonekedwe a ziwengo - khungu ndi kupuma (mpaka edema la Quincke kapena bronchospasm)
  • Aspirin anapambana
  • Matenda a Stool, kupweteka kwam'mimba, kutuluka kwamkati, kutaya mtima
  • Kuwonongeka kwa impso
  • Mpweya kutulutsa magazi, mphuno zam'mimba, kuwonda komanso kusokonezeka kwa magazi.

Ngati pali zizindikiro zokayikitsa mutatha kutenga Aspirin Oops, ziyenera kuchotsedwa ndikuyang'ana kwa dokotala.

Mlingo wa Aspirin Oops

Makampani opanga mankhwala amapanga Aspirin Oops, womwe ndi phale loyera, lathyathyathya. Mapiritsi ali ndi 500 mg yogwira ntchito - acetylsalicylic acid. Aspirin Oops amakhalanso opeza. Izi ndi sodium carbonate, citric acid, sodium citrate. Kuphatikizika kwa mankhwalawa kumakhalanso ndi sodium bicarbonate, aspartame, flavorings. Phukusili limakhala ndi miyala inayi ya Aspirin Oops.

Aspirin Oops effeedcent mapiritsi alinso 325 mg wa acetylsalicylic acid.

Mlingo ndi kasamalidwe ka Aspirin Oops

Malinga ndi malangizo, Aspirin Oops amatengedwa pakamwa, 500-1000 mg patsiku. Mulingo wambiri watsiku ndi tsiku wa Aspirin Oops ukhoza kukhala magalamu atatu. Nthawi zambiri mankhwala amagwiritsidwa ntchito kamodzi kapena kawiri patsiku, katatu angagwiritsidwe ntchito. Musanagwiritse ntchito, piritsi la mankhwala liyenera kusungunuka mu kapu yamadzi. Ngati kupweteka kwambiri kumakhala kovuta ndipo pamakhala kutentha kwambiri kumayambiriro kwa matendawa, ndiye kuti mutha kumwa mapiritsi awiri nthawi imodzi. Tsiku kuti musamamwe zosaposera zisanu ndi chimodzi. Akuluakulu amalangizidwa kuti asatenge mapiritsi anayi a Aspirin Oops. Monga antipyretic, Aspirin Oops amatengedwa kwa masiku atatu, monga analgesic, mutha kutenga masiku asanu.

Ana osakwana zaka zinayi ali osavomerezeka kuti azipereka Aspirin Oops. Kuyambira wazaka 4 mpaka 6 zimapatsa 200 mg patsiku, zaka 7-9 zimatenga 300 mg tsiku lililonse. Ana opitirira zaka 12 amatha kumwa 250 mg kawiri pa tsiku, pomwe mlingo wa tsiku ndi tsiku sayenera kupitirira 750 mg.

Ndi kulowetsedwa kwa myocardial, odwala amatha kutenga Aspirin Oops kuchokera 40 mpaka 325 mg kamodzi patsiku. Mankhwala amagwiritsidwanso ntchito ngati choletsa chophatikizira cha kupatsidwa zinthu za m'magazi. Pankhaniyi, Aspirin Oops amatengedwa pa mlingo wa 325 mg tsiku lililonse kwa nthawi yayitali.

Kuchita ndi mankhwala ena

Malinga ndi malangizo, Aspirin Oops imatha kupititsa patsogolo zotsatira za heparin ndi anticoagulants pamlomo, komanso ma reserpine, mahomoni a steroid. Mankhwala amachepetsa mphamvu ya mankhwala a antihypertensive mukamawagwiritsa ntchito. Kugwiritsa ntchito kwa Aspirin Oops ndi mankhwala ena omwe si a antiidal komanso anti-yotupa kumatha kubweretsa zovuta zoyipa.

Migwirizano ndi magwiritsidwe akusungidwa

Chogulacho ndi choyenera kugwiritsidwa ntchito patatha zaka zitatu kuyambira tsiku lomwe amatulutsa. Pofuna kupewa kutayika kwa mankhwala othandizira, ayenera kutetezedwa kuti asatenthedwe, kuwala komanso kutentha kwambiri. Sungani kutentha mpaka 25 ° C, khalani kutali ndi ana.

Kusankha malonda okhala ndi acetylsalicylic acid si vuto masiku ano. Koma potengera mawonekedwe ake a pharmacological, kusinthaku kuyenera kuchitika mothandizidwa ndi dokotala.

Bayer (Germany)

Mtengo wapakati: 258 rub

Chogulitsachi chili ndi 400 mg yogwira ntchito, yopatsidwa vitamini C (240 mg). Zowonjezera ndi zosakaniza zomwe zimapanga kapangidwe kake ndi kusinthasintha kwa mankhwalawo. Mankhwalawa amapezeka mu mawonekedwe a mapiritsi akulu oyera pokonzekera chakumwa, kumbali ina pali chizindikiro cha lingaliro la nkhawa.

Mankhwala amatengedwa piritsi limodzi kusungunuka m'madzi, muyeso wovomerezeka umodzi ndi mapiritsi awiri, mlingo wachiwiri pambuyo maola anayi.

Ubwino:

  • Khalidwe labwino kwambiri
  • Kachitidwe.

Zoyipa:

  • Zomwe zimachitika sizingachitike.

Kusiya Ndemanga Yanu